Peptidomimetics Protocols
In Peptidomimetics Protocols, Wieslaw Kazmierski assembles a state-of-the-art collection of detailed synthetic procedures that lead to a variety of scaffolds, turn mimetics, peptide-bond replacements, and enzyme inhibitors. Topics range from syntheses of unusual amino acids, to the use of a variety...
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| Format: | eBook |
| Language: | English |
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Totowa, NJ
Humana Press
1999, 1999
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| Edition: | 1st ed. 1999 |
| Series: | Methods in Molecular Medicine
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| Subjects: | |
| Online Access: | |
| Collection: | Springer Protocols Archive 1981-2004 - Collection details see MPG.ReNa |
Table of Contents:
- Synthesis and Use of Pseudopeptides Derived from 1,2,4-Oxadiazole-, 1,3,4-Oxadiazole-, and 1,2,4-Triazole-based Dipeptidomimetics
- Synthesis of Aminobenzoic Acid-Based Nonpeptide Templates: Applications in Peptidomimetic Drug Discovery
- Synthesis of an Esterase-Sensitive Cyclic Prodrug of a Model Hexapeptide Having Enhanced Membrane Permeability and Enzymatic Stability Using an Acyloxyalkoxy Promoiety
- Synthesis of an Esterase-Sensitive Cyclic Prodrug of a Model Hexapeptide Having Enhanced Membrane Permeability and Enzymatic Stability Using a 3-(2?-Hydroxy-4?,6?-Dimethylphenyl)-3,3-Dimethyl Propionic Acid Promoiety
- Synthesis of Coumarin-Based, Esterase-Sensitive Cyclic Prodrugs of Opioid Peptides with Enhanced Membrane Permeability and Enzymatic Stability
- Azatides as Peptidomimetics: Solution and Liquid Phase Syntheses
- Synthesis of Cbz-Protected Ketomethylene Dipeptide Isosteres
- (E)-Alkene Peptide Bond Isosteres by Cuprate Opening of Vinyl Aziridines
- Synthesis of 3-Amino-l-CarboxymethyI-Benzodiazepine (BZA) Peptidomimetics
- A Conformationally Restricted ?-Strand HIV Protease Inhibitor
- Synthesis of Cyclopropane-Containing Leu-Enkephalin Analogs
- The 1,5-Disubstituted Tetrazole Ring as a cis-Amide Bond Surrogate
- Synthesis of (2R, 3R, 4R, 5S)-5-tert-Butyloxycarbonylamino-3,4-Dihydroxy-2-1sopropyl-3,4-O,O-Isopropylidene-6-CyctohexyI-Hexanoic Acid
- Synthesis of (2S, 4S, 5S)-5-(t-Butoxycarbonylamino)-4-(t-Butyldimethylsilyloxy)-2-Isopropyl-7-Methyl Octanoic Acid
- Synthesis of ?-Vinyl Amino Acids
- A Novel Synthetic Protocol for the Preparation of Enantiopure 3-, 4-, and 5-Substituted Prolines
- Synthesis of Aminobenzoic Acid-Based Nonpeptide Templates
- Aminimides as Peptidomimetics
- Syntheses of Norstatine, Its Analogs, and Dipeptide Isosteres by Means of ?-Lactam Synthon Method
- Synthesis of a Versatile Peptidomimetic Scaffold
- An Asymmetric Synthesis Protocol to Prepare Topographically Constrained ?-Substituted Aromatic Amino Acids
- Synthesis of Oligopeptides Containing an Oxirane Ring in the Place of a Peptidic Bond
- Synthesis of Protected Lactam-Bridged Dipeptides
- Synthesis of Peptidomimics Through Sugar-Based Scaffolds
- The Synthesis of Bicyclic Piperazinone and Related Derivatives
- Synthesis of Dipeptides with ?[CH20] Amide Bond Mimetics
- SNAr-Based Cycloetherification Methodology: Application in the Synthesis of Heterodectic Macrocyclic Peptides with Endo Aryl-Aryl and Aryl-Alkyl Ether Bonds
- Cyclic Aromatic Amino Acids with Constrained ?1 and ?2 Dihedral Angles
- Asymmetric Syntheses of Unnatural Amino Acids and Hydroxyethylene Peptide Isosteres
- Fluoroolefin Isosteres